Brivudine

Brivudine

SCHEMBL4283382

O=c1[nH]c(=O)n(C2CC(O)C(CO)O2)cc1/C=C/Br

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TK1 P04183 4/20 1.00
CYP1A2 P05177 1/20 1.00
CYP3A4 P08684 1/20 1.00
TSHR P16473 1/20 1.00
BLM P54132 1/20 1.00
PMP22 Q01453 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
LMNA P02545 2/20 0.66
SMN1; SMN2 Q16637 2/20 0.66
TK2 O00142 5/20 0.65
ALOX12 P18054 1/20 0.62
ADRA1A P35348 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Brivudine SCHEMBL13030272 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL4283383 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL4314668 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL141407 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL13674189 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL1172398 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL99350 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL5983819 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL21316784 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL15405329 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11786541-B2 Inhibitor of sphingosine kinase 2 for treating Ebola REDHILL BIOPHARMA LTD. (IL) 2023-10-17 US disclosed
US-11786541-B2 Inhibitor of sphingosine kinase 2 for treating Ebola REDHILL BIOPHARMA LTD. (IL) 2023-10-17 US disclosed
US-20210369754-A1 INHIBITOR OF SPHINGOSINE KINASE 2 FOR TREATING EBOLA REDHILL BIOPHARMA LTD (IL) 2021-12-02 US disclosed
US-11090325-B2 Compositions for treating ebola virus infection REDHILL BIOPHARMA LTD. (IL) 2021-08-17 US disclosed
US-10946000-B2 Method for treating cancer with combination therapy REDHILL BIOPHARMA LTD. (IL) 2021-03-16 US disclosed
US-20200155585-A1 COMPOSITIONS FOR TREATING EBOLA VIRUS INFECTION REDHILL BIOPHARMA LTD (IL) 2020-05-21 US disclosed
US-10543222-B2 Therapy for inhibition of single-stranded RNA virus replication REDHILL BIOPHARMA LTD. (IL) 2020-01-28 US disclosed
US-10463654-B2 Combination therapies for treating cancer REDHILL BIOPHARMA LTD. (IL) 2019-11-05 US disclosed
US-9974800-B2 Therapy for inhibition of single-stranded RNA virus replication REDHILL BIOPHARMA LTD. (IL) 2018-05-22 US disclosed
US-9974800-B2 Therapy for inhibition of single-stranded RNA virus replication REDHILL BIOPHARMA LTD. (IL) 2018-05-22 US disclosed
US-20130210757-A1 DOUBLE-LIVER-TARGETING PHOSPHORAMIDATE AND PHOSPHONOAMIDATE PRODRUGS NANJING MOLECULAR RESEARCH, INC. (CN) 2013-08-15 US disclosed
EP-1898935-B1 NORTH-2'-DEOXY-METHANOCARBATHYMIDINES AS ANTIVIRAL AGENTS AGAINST POXVIRUSES US GOV HEALTH & HUMAN SERV (US) 2012-09-19 EP disclosed
US-7951787-B2 Phosphoramidate compounds and methods of use CARDIFF PROTIDES LIMITED (GB) 2011-05-31 US disclosed
US-7951787-B2 Phosphoramidate compounds and methods of use CARDIFF PROTIDES LIMITED (GB) 2011-05-31 US disclosed
WO-2009129094-A2 COMPOSITIONS CONTAINING ANTIVIRAL COMPOUNDS AND METHODS OF USING THE SAME MALLINCKRODT INC. (US) 2009-10-22 WO disclosed
US-20090258843-A1 Compositions Containing Antiviral Compounds and Methods of Using the Same MALLINCKRODT INC. (US) 2009-10-15 US disclosed
US-20090258843-A1 Compositions Containing Antiviral Compounds and Methods of Using the Same MALLINCKRODT INC. (US) 2009-10-15 US disclosed
US-20090258843-A1 Compositions Containing Antiviral Compounds and Methods of Using the Same MALLINCKRODT INC. (US) 2009-10-15 US disclosed
US-20090221523-A1 North-2'-deoxy-methanocarbathymidines as antiviral agents against poxviruses HEALTH AND HUMAN SERVICES, THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF 2009-09-03 US disclosed
US-20090221523-A1 North-2'-deoxy-methanocarbathymidines as antiviral agents against poxviruses HEALTH AND HUMAN SERVICES, THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF 2009-09-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090258843-A1 Compositions Containing Antiviral Compounds and Methods of Using the Same EIF2AK2, MAVS, IRF3 TK1 732/4885CYP1A2 3115/4885CYP3A4 1281/4885
US-10543222-B2 Therapy for inhibition of single-stranded RNA virus replication RNMT, EIF2AK2, POLRMT TK1 451/4885CYP1A2 4681/4885CYP3A4 4538/4885
US-11786541-B2 Inhibitor of sphingosine kinase 2 for treating Ebola SPHK2, SPHK1, S1PR2 TK1 385/4885CYP1A2 4267/4885CYP3A4 4417/4885
US-20200155585-A1 COMPOSITIONS FOR TREATING EBOLA VIRUS INFECTION NEFM, EIF2AK2, IRF3 TK1 1425/4885CYP1A2 4500/4885CYP3A4 4212/4885
US-20090221523-A1 North-2'-deoxy-methanocarbathymidines as antiviral agents against poxviruses SAMHD1, TK2, DCTD TK1 62/4885CYP1A2 1717/4885CYP3A4 2432/4885
US-10946000-B2 Method for treating cancer with combination therapy TPMT, KRAS, SDHA TK1 1878/4885CYP1A2 344/4885CYP3A4 239/4885
US-20130210757-A1 DOUBLE-LIVER-TARGETING PHOSPHORAMIDATE AND PHOSPHONOAMIDATE PRODRUGS PNP, PAICS, NTPCR TK1 34/4885CYP1A2 1048/4885CYP3A4 922/4885
US-20210369754-A1 INHIBITOR OF SPHINGOSINE KINASE 2 FOR TREATING EBOLA SPHK2, SPHK1, S1PR2 TK1 385/4885CYP1A2 4267/4885CYP3A4 4417/4885
US-10463654-B2 Combination therapies for treating cancer TPMT, KRAS, ACE TK1 2512/4885CYP1A2 437/4885CYP3A4 199/4885
US-11090325-B2 Compositions for treating ebola virus infection NEFM, EIF2AK2, IRF3 TK1 1425/4885CYP1A2 4500/4885CYP3A4 4212/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.