SCHEMBL8294430

SCHEMBL8294430

COC(=O)C1Cc2ccncc2CN1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD17B10 Q99714 1/20 0.44
NAMPT P43490 1/20 0.39
ROCK2 O75116 1/20 0.36
DPP4 P27487 1/20 0.35
GLA P06280 1/20 0.35
HDAC8 Q9BY41 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
BLM P54132 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8294431 0.94 KDM4E (0.44) KDM4EALDH1A1GAACYP1A2CYP2D6
SCHEMBL6254144 0.82 EGLN1 (0.44) KDM4EALDH1A1GAAMAPTHSD17B10
SCHEMBL1491698 0.80 KDM4E (0.56) KDM4EALDH1A1GAACYP1A2CYP2D6
SCHEMBL1491696 0.80 KDM4E (0.56) KDM4EALDH1A1GAACYP1A2CYP2D6
SCHEMBL32677077 0.80 KDM4E (0.56) KDM4EALDH1A1GAACYP1A2CYP2D6
SCHEMBL6866846 0.80 KDM4E (0.56) KDM4EALDH1A1GAACYP1A2CYP2D6
SCHEMBL29707282 0.80 KDM4E (0.56) KDM4EALDH1A1GAACYP1A2CYP2D6
SCHEMBL29715383 0.80 KDM4E (0.56) KDM4EALDH1A1GAACYP1A2CYP2D6
SCHEMBL13604128 0.79 NAMPT (0.42) KDM4EALDH1A1GAACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL30665771 0.79 KDM4E (0.55) KDM4EALDH1A1GAACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005056013-A1 DPP-IV INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) GMBH (CH) 2005-06-23 WO disclosed