SCHEMBL8294455

SCHEMBL8294455

CC(=O)NC1(C)CC2CCCN(Cc3ccccc3)C2C1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.42
NPSR1 Q6W5P4 1/20 0.40
NPY1R P25929 1/20 0.39
HTT P42858 1/20 0.39
NPY2R P49146 1/20 0.39
HSD11B1 P28845 2/20 0.39
SLC18A3 Q16572 1/20 0.39
OPRD1 P41143 1/20 0.38
CCR2 P41597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8293267 0.79 NPY1R (0.47) SIGMAR1NPY1RHTTNPY2RSLC18A3
SCHEMBL21653769 0.74 KMT2A (0.46) OPRD1
SCHEMBL2851430 0.74 KMT2A (0.46) OPRD1
SCHEMBL21631693 0.74 KMT2A (0.46) OPRD1
SCHEMBL2851436 0.74 KMT2A (0.46) OPRD1
SCHEMBL12836223 0.73 NPY1R (0.52) SIGMAR1NPY1RHTTNPY2RSLC18A3
SCHEMBL1991966 0.70 CYP2D6 (0.59) SIGMAR1
SCHEMBL12836641 0.70 NPY1R (0.43) SIGMAR1NPY1RHTTNPY2RSLC18A3
SCHEMBL1318062 0.70 LTA4H (0.52) SIGMAR1NPY1RHTTNPY2R
SCHEMBL14598757 0.69 NPSR1 (0.55) NPSR1HSD11B1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664031-B1 ADAMANTANE AND AZABICYCLO-OCTANE AND NONANE DERIVATIVES PROCESS OF THEIR PREPARATION AND THEIR USE AS DPP-IV INHIBITORS SANOFI AVENTIS (FR) 2007-12-19 EP disclosed
WO-2005021536-A2 ADAMANTANE AND AZABICYCLO-OCTANE AND NONANE DERIVATIVES, PROCESS OF THEIR PREPARATION AND THEIR USE AS DPP-IV INHIBITORS SANOFI-AVENTIS (FR) 2005-03-10 WO disclosed