SCHEMBL8294589

SCHEMBL8294589

CC1C(=O)CN(Cc2ccccc2)CC1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.53
SIGMAR1 Q99720 2/20 0.50
GAA P10253 1/20 0.50
MC4R P32245 1/20 0.47
LMNA P02545 2/20 0.46
POLB P06746 1/20 0.46
TACR1 P25103 2/20 0.45
FUCA1 P04066 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
KMT2A Q03164 1/20 0.44
F2 P00734 1/20 0.44
PLG P00747 1/20 0.44
ELANE P08246 1/20 0.44
CTSG P08311 1/20 0.44
CMA1 P23946 1/20 0.44
CTRC Q99895 1/20 0.44
CCR3 P51677 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9379752 0.82 ACHE (0.50) ACHESIGMAR1GAAMC4RLMNA
SCHEMBL19261315 0.81 CYP2D6 (0.47) ACHESIGMAR1GAAMC4RFUCA1
SCHEMBL5766167 0.80 ACHE (0.60) ACHESIGMAR1MC4RCCR3
SCHEMBL9583954 0.80 ABL1 (0.49) ACHESIGMAR1GAAFUCA1KDM4E
SCHEMBL692536 0.80 ACHE (0.60) ACHESIGMAR1MC4RCCR3
SCHEMBL1105751 0.80 ACHE (0.60) ACHESIGMAR1MC4RCCR3
SCHEMBL23580062 0.79 TSHR (0.44) ACHEPOLBALDH1A1KMT2A
Hydrochloric Acid SCHEMBL28093485 0.78 ACHE (0.58) ACHESIGMAR1TACR1CCR3
SCHEMBL2438031 0.78 SIGMAR1 (0.60) ACHESIGMAR1GAAMC4RLMNA
SCHEMBL30881357 0.77 ACHE (0.45) ACHESIGMAR1GAAMC4RTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005013914-A2 HETEROARYLAMINOSULFONYLPHENYL DERIVATIVES FOR USE AS SODIUM OR CALCIUM CHANNEL BLOCKERS IN THE TREATMENT OF PAIN VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-02-17 WO disclosed