SCHEMBL8299997

SCHEMBL8299997

C=Cc1cc(O)c(O)c(Br)c1Br

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.46
IGF1R P08069 2/20 0.41
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA4 P22748 3/20 0.38
CA6 P23280 3/20 0.38
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
RECQL P46063 1/20 0.33
HIF1A Q16665 1/20 0.33
HSD17B10 Q99714 1/20 0.33
AKR1B1 P15121 1/20 0.31
TNKS O95271 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8996046 0.77 ERN1 (0.47) PTPN1IGF1R
SCHEMBL29446638 0.77 ERN1 (0.47) PTPN1IGF1R
SCHEMBL2817418 0.73 ESR2 (0.33) ESR1ESR2
SCHEMBL29420749 0.73 ESR2 (0.33) ESR1ESR2
SCHEMBL23516391 0.72 XDH (0.37) ESR1ESR2ALDH1A1HPGDAKR1B1
SCHEMBL27925993 0.70 PRKCG (0.31) ESR1ESR2
SCHEMBL9571705 0.70 POLB (0.35) ESR1ESR2ALDH1A1ALOX15
SCHEMBL31132199 0.69 PTPN1 (0.38) PTPN1IGF1RCA1CA2CA4
SCHEMBL40037 0.69 EIF2AK2 (0.47) AKR1B1
SCHEMBL27773344 0.69 PTPN1 (0.52) PTPN1CA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037779-A2 NOVEL DIPEPTIDYL PEPTIDASE IV INHIBITORS USED FOR FUNCTIONALLY INFLUENCING DIFFERENT CELLS AND TREATING IMMUNOLOGICAL, INFLAMMATORY, NEURONAL, AND OTHER DISEASES IMTM GMBH (DE) 2005-04-28 WO disclosed