SCHEMBL8300063

SCHEMBL8300063

CC(=O)c1ccc(-c2ccc(-c3csc(C(=O)N[C@H](CC(=O)O)c4ccccc4)c3)cc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 9/20 0.76
MMP13 P45452 3/20 0.76
MMP3 P08254 1/20 0.76
MMP9 P14780 1/20 0.76
MMP8 P22894 1/20 0.76
AKT1 P31749 5/20 0.46
ROCK1 Q13464 4/20 0.46
RPS6KA5 O75582 3/20 0.46
GSK3B P49841 3/20 0.46
NEK4 P51957 3/20 0.46
PRKCD Q05655 3/20 0.46
PRKG2 Q13237 3/20 0.46
PRKG1 Q13976 3/20 0.46
PKN2 Q16513 3/20 0.46
CLK4 Q9HAZ1 3/20 0.46
ROCK2 O75116 3/20 0.46
MAPK13 O15264 2/20 0.46
MAP4K4 O95819 2/20 0.46
PRKCG P05129 2/20 0.46
CDK1 P06493 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6367846 1.00 MMP12 (0.76) MMP12MMP13MMP3MMP9MMP8
SCHEMBL4321262 0.86 MMP12 (1.00) MMP12MMP13MMP3MMP9MMP8
SCHEMBL8298104 0.86 MMP12 (1.00) MMP12MMP13MMP3MMP9MMP8
Hydrochloric Acid SCHEMBL6662154 0.85 MMP12 (0.98) MMP12MMP13MMP3MMP9MMP8
SCHEMBL6368918 0.83 MMP12 (0.74) MMP12MMP13MMP3MMP9MMP8
SCHEMBL6369477 0.83 MMP12 (0.74) MMP12MMP13MMP3MMP9MMP8
SCHEMBL6367899 0.81 MMP12 (0.73) MMP12MMP13MMP3MMP9MMP8
SCHEMBL6370866 0.81 MMP12 (1.00) MMP12MMP13MMP3MMP9MMP8
SCHEMBL8301127 0.80 MMP12 (0.57) MMP12MMP13MMP3MMP9MMP8
SCHEMBL6367844 0.78 MMP12 (0.51) MMP12MMP13MMP3MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003115-A1 THIOPHENE AMINO ACID DERIVATIVES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM WARNER-LAMBERT COMPANY LLC (US) 2005-01-13 WO disclosed