SCHEMBL8300077

SCHEMBL8300077

c1cc(NCCCN2CCNCC2)ccn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.56
CYP2D6 P10635 2/20 0.56
KDR P35968 1/20 0.45
SIGMAR1 Q99720 2/20 0.44
CYP2C19 P33261 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
ALDH1A1 P00352 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
ADRB2 P07550 1/20 0.42
NCF1 P14598 1/20 0.42
PLD1 Q13393 1/20 0.42
ROCK1 Q13464 2/20 0.39
PRKCZ Q05513 1/20 0.39
ACP1 P24666 1/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304884 0.90 CYP3A4 (0.63) CYP3A4CYP2D6KDRSIGMAR1L3MBTL1
SCHEMBL6649060 0.85 HRH3 (0.51) CYP3A4CYP2D6CYP2C19L3MBTL1ACP1
SCHEMBL6651015 0.84 CYP3A4 (0.53) CYP3A4CYP2D6CYP2C19L3MBTL1ACP1
SCHEMBL6649751 0.81 CYP2C19 (0.65) CYP3A4CYP2D6CYP2C19L3MBTL1ALDH1A1
SCHEMBL14409559 0.78 CYP3A4 (0.46) CYP3A4CYP2D6CYP2C19L3MBTL1
SCHEMBL23657189 0.76 CA1 (0.63) ALDH1A1KDM4ECA1CA2CA9
SCHEMBL1509423 0.76 SIGMAR1 (0.70) CYP3A4CYP2D6SIGMAR1L3MBTL1ADRB2
SCHEMBL2127950 0.75 HRH3 (0.55) CYP3A4CYP2D6SIGMAR1L3MBTL1
SCHEMBL30341164 0.74 SIGMAR1 (0.63) CYP3A4CYP2D6SIGMAR1L3MBTL1
SCHEMBL7672095 0.73 SIGMAR1 (0.53) CYP3A4CYP2D6KDRSIGMAR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed
US-5786371-A INHIBIT AGGREGATION OF BLOOD PLATELETS BOEHRINGER MANNHEIM GMBH (DE) 1998-07-28 US disclosed
EP-0808306-A1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1997-11-26 EP disclosed
WO-1996024586-A1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1996-08-15 WO disclosed