SCHEMBL8300346

SCHEMBL8300346

COc1cccc(C[N+]2([O-])CCCC(CCCN3CCC(O)(c4ccccc4)CC3)(c3ccc(Cl)c(Cl)c3)C2)c1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 10/20 0.45
TACR2 P21452 9/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
KMT2A Q03164 1/20 0.43
TACR3 P29371 6/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8742822 0.99 TACR1 (0.45) TACR1TACR2MEN1ALDH1A1LMNA
SCHEMBL8300821 0.84 SLC6A4 (0.37) TACR1TACR2CYP2D6
SCHEMBL7313003 0.83 TACR1 (0.55) TACR1TACR2MEN1ALDH1A1LMNA
Hydrochloric Acid SCHEMBL8742497 0.82 TACR1 (0.54) TACR1TACR2MEN1ALDH1A1LMNA
SCHEMBL8292836 0.79 TACR2 (0.34) TACR1TACR2TACR3CYP2D6
SCHEMBL8300343 0.77 TACR1 (0.75) TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL8742817 0.77 TACR1 (0.74) TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL8592981 0.74 TACR1 (0.51) TACR1TACR2MEN1ALDH1A1LMNA
SCHEMBL8300818 0.73 CCR5 (0.43) TACR1ALDH1A1
Hydrochloric Acid SCHEMBL8521991 0.72 CCR5 (0.42) TACR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP disclosed
US-5625060-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions on which they are present Sanofi, Elf (FR) 1997-04-29 US disclosed
US-5340822-A Substance P, neurokinin antagonists ELF SANOFI (FR) 1994-08-23 US disclosed
EP-0512901-A1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI (FR) 1992-11-11 EP disclosed