SCHEMBL8300818

SCHEMBL8300818

[O-][N+]1(Cc2ccccc2)CCCC(CCN2CCC(Cc3ccccc3)CC2)(c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.43
SLC6A2 P23975 5/20 0.41
SLC6A4 P31645 5/20 0.41
TACR1 P25103 5/20 0.41
CCR3 P51677 2/20 0.40
SLC6A3 Q01959 2/20 0.40
NPFFR1 Q9GZQ6 1/20 0.40
NPFFR2 Q9Y5X5 1/20 0.40
PRMT3 O60678 1/20 0.39
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
PRMT1 Q99873 1/20 0.39
PRMT8 Q9NR22 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8521991 0.99 CCR5 (0.42) CCR5SLC6A2SLC6A4TACR1CCR3
SCHEMBL8296371 0.81 SLC6A2 (0.43) CCR5SLC6A2SLC6A4TACR1CCR3
SCHEMBL8300496 0.80 SLC6A2 (0.54) CCR5SLC6A2SLC6A4TACR1CCR3
Hydrochloric Acid SCHEMBL8742517 0.79 SLC6A2 (0.53) CCR5SLC6A2SLC6A4TACR1CCR3
SCHEMBL8296084 0.78 CCR5 (0.64) CCR5TACR1
Hydrochloric Acid SCHEMBL8522900 0.77 CCR5 (0.63) CCR5TACR1
SCHEMBL8296368 0.75 TACR1 (0.50) CCR5TACR1
SCHEMBL8300814 0.74 TACR1 (0.73) CCR5TACR1
SCHEMBL8296292 0.73 SLC6A4 (0.36) SLC6A2SLC6A4TACR1SLC6A3
Hydrochloric Acid SCHEMBL8521990 0.73 TACR1 (0.72) CCR5TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999007413-A1 SUBSTANCE P INHIBITORS IN COMBINATION WITH NMDA-BLOCKERS FOR TREATING PAIN ALGOS PHARMACEUTICAL CORPORATION (US) 1999-02-18 WO claimed
JP-5186425-A None JP disclosed
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP disclosed
JP-H05186425-A POLYCYCLIC AMINE COMPOUND, ITS ENANTIOMER, ITS PREPARATION AND PHARMACEUTIC COMPOSITION CONTAINING THOSE ELF SANOFI 1993-07-27 JP disclosed
EP-0512901-A1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI (FR) 1992-11-11 EP disclosed