SCHEMBL8300679

SCHEMBL8300679

O=C(O)CC1CCC(C2CCN(CCCNc3ccncc3)CC2)CC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 5/20 0.39
CYP2D6 P10635 2/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
CYP2C9 P11712 1/20 0.38
GRIN2B Q13224 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A3 Q01959 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300003 0.97 CCR3 (0.39) CCR3CYP2D6ITGB3ITGA2BCYP2C9
SCHEMBL8302166 0.93 ITGB3 (0.39) CYP2D6ITGB3ITGA2BCYP2C9GRIN2B
SCHEMBL8300507 0.88 KDM4E (0.43) CYP2D6ITGB3ITGA2B
SCHEMBL8304879 0.84 KDM4E (0.42) CCR3CYP2D6ITGB3ITGA2BCYP2C9
SCHEMBL8300030 0.81 KDM4E (0.45) CYP2D6ITGB3ITGA2BCYP2C9GRIN2B
SCHEMBL8302338 0.78 ITGB3 (0.42) CYP2D6ITGB3ITGA2BCYP2C9GRIN2B
SCHEMBL8300686 0.76 NAMPT (0.43) CYP2D6ITGB3ITGA2BCYP2C9GRIN2B
SCHEMBL8298652 0.74 ITGB3 (0.45) CYP2D6ITGB3ITGA2BCYP2C9GRIN2B
SCHEMBL8615084 0.74 ITGB3 (0.37) CYP2D6ITGB3ITGA2BCYP2C9GRIN2B
SCHEMBL6649060 0.74 HRH3 (0.51) CYP2D6CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed
EP-0808306-A1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1997-11-26 EP disclosed
WO-1996024586-A1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1996-08-15 WO disclosed