SCHEMBL8300507

SCHEMBL8300507

O=C(O)CC1CCC(N2CCN(CCCNc3ccncc3)CC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
TRPV6 Q9H1D0 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
L3MBTL3 Q96JM7 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304879 0.97 KDM4E (0.42) KDM4EMEN1ALDH1A1KMT2ATRPV6
SCHEMBL8300030 0.93 KDM4E (0.45) KDM4EMEN1ALDH1A1KMT2ATRPV6
SCHEMBL8300679 0.88 CCR3 (0.39) CYP2D6ITGB3ITGA2B
SCHEMBL8304380 0.85 DRD3 (0.36) KDM4EMEN1ALDH1A1KMT2ATRPV6
SCHEMBL8300686 0.85 NAMPT (0.43) KDM4EMEN1ALDH1A1KMT2ATRPV6
SCHEMBL8300003 0.84 CCR3 (0.39) CYP2D6ITGB3ITGA2B
SCHEMBL8298652 0.83 ITGB3 (0.45) KDM4EMEN1ALDH1A1KMT2ATRPV6
SCHEMBL8299936 0.82 KDM4E (0.41) KDM4EMEN1ALDH1A1KMT2ATRPV6
SCHEMBL8318264 0.82 DRD2 (0.47) TRPV6ITGB3ITGA2B
SCHEMBL8305139 0.82 CDK9 (0.36) KDM4EMEN1ALDH1A1KMT2ATRPV6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed