SCHEMBL8300768

SCHEMBL8300768

CC(C)Oc1cccc(CC(=O)N2CCCC(CCN3CCC(Cc4ccccc4)CC3)(c3ccc(Cl)c(Cl)c3)C2)c1

nearest known ligand 0.70

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 2/20 0.69
TACR1 P25103 2/20 0.69
CCR5 P51681 1/20 0.55
HRH1 P35367 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8296084 0.89 CCR5 (0.64) TACR2TACR1CCR5
Hydrochloric Acid SCHEMBL8522900 0.89 CCR5 (0.63) TACR2TACR1CCR5
SCHEMBL8296058 0.88 TACR2 (0.54) TACR2TACR1CCR5
SCHEMBL9027933 0.88 TACR1 (0.65) TACR2TACR1CCR5HRH1
SCHEMBL9027942 0.88 TACR1 (0.65) TACR2TACR1CCR5HRH1
Hydrochloric Acid SCHEMBL8591404 0.88 TACR2 (0.53) TACR2TACR1CCR5
SCHEMBL9032557 0.87 TACR1 (0.65) TACR2TACR1CCR5HRH1
SCHEMBL9028482 0.87 TACR1 (0.65) TACR2TACR1CCR5HRH1
SCHEMBL9028476 0.87 TACR1 (0.65) TACR2TACR1CCR5HRH1
SCHEMBL9028136 0.87 TACR1 (0.65) TACR2TACR1CCR5HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP disclosed
US-5625060-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions on which they are present Sanofi, Elf (FR) 1997-04-29 US disclosed
US-5340822-A Substance P, neurokinin antagonists ELF SANOFI (FR) 1994-08-23 US disclosed
EP-0512901-A1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI (FR) 1992-11-11 EP disclosed