SCHEMBL8300808

SCHEMBL8300808

Cc1cn([C@H]2C[C@H](C(=O)O)N(C(=O)OC(C)(C)C)C2)c(=O)[nH]c1=O

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TK1 P04183 3/20 0.39
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
P2RX3 P56373 1/20 0.37
PARP1 P09874 1/20 0.37
HSD11B1 P28845 1/20 0.37
RNASE1 P07998 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8646363 1.00 TK1 (0.39) TK1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL8298155 1.00 TK1 (0.39) TK1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL8304127 1.00 TK1 (0.39) TK1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL8303221 0.86 CYP1A2 (0.39) TK1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL8298156 0.85 TK1 (0.38) TK1PARP1HSD11B1RNASE1
SCHEMBL8304128 0.85 TK1 (0.38) TK1PARP1HSD11B1RNASE1
SCHEMBL8300811 0.85 TK1 (0.38) TK1PARP1HSD11B1RNASE1
SCHEMBL13956884 0.78 DRD2 (0.37) TK1RNASE1
SCHEMBL8304914 0.72 SRC (0.43)
SCHEMBL8639265 0.72 SRC (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0646596-B1 Nucleic acid binding oligomers having C-branches for therapy and diagnosis BAYER AG (DE) 1999-05-26 EP disclosed
US-5849893-A Nucleic acid-binding oligomers possessing C-branching for therapy and diagnostics BAYER AKTIENGESELLSCHAFT (DE) 1998-12-15 US disclosed
EP-0646596-A1 Nucleic acid binding oligomers having C-branches for therapy and diagnosis BAYER AG (DE) 1995-04-05 EP disclosed