SCHEMBL8301717

SCHEMBL8301717

N#CCCCc1cccc2cc[nH]c12

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.41
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MPO P05164 1/20 0.38
SLC6A4 P31645 1/20 0.38
KEAP1 Q14145 1/20 0.37
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
PDPK1 O15530 1/20 0.36
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306159 0.90 AHR (0.43) AHRKEAP1HTR2AHTR2CPDPK1
SCHEMBL2261191 0.81 AHR (0.47) AHRKEAP1PDPK1BACE1
SCHEMBL31561732 0.78 AHR (0.44) AHRKEAP1HTR2AHTR2CPDPK1
SCHEMBL3790923 0.78 AHR (0.44) AHRKEAP1HTR2AHTR2CPDPK1
SCHEMBL28362482 0.78 AHR (0.44) AHRKEAP1HTR2AHTR2CPDPK1
SCHEMBL6029507 0.78 AHR (0.44) AHRKEAP1HTR2AHTR2CPDPK1
SCHEMBL31561738 0.78 AHR (0.44) AHRKEAP1HTR2AHTR2CPDPK1
SCHEMBL9248977 0.77 AHR (0.43) AHRKEAP1HTR2AHTR2C
SCHEMBL2260654 0.77 MPO (0.46) AHRMPOSLC6A4KEAP1HTR2A
SCHEMBL9026320 0.75 AHR (0.42) AHRKEAP1HTR2AHTR2CPDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469833-B1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY CO ELI (GB) 1999-09-08 EP disclosed
US-5281593-A Pharmaceuticals LILLY INDUSTRIES LIMITED (GB) 1994-01-25 US disclosed
EP-0469833-A1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY INDUSTRIES LIMITED (GB) 1992-02-05 EP disclosed