SCHEMBL8301724

SCHEMBL8301724

COc1nc(-c2ccc(OC(F)(F)F)cc2)cc2cc(N(C)C)ccc12

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 2/20 0.50
ADORA3 P0DMS8 1/20 0.40
F2RL3 Q96RI0 1/20 0.39
MAT2A P31153 1/20 0.39
TLR9 Q9NR96 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
PTGDR Q13258 1/20 0.38
DHODH Q02127 1/20 0.38
APP P05067 1/20 0.38
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
SCN5A Q14524 3/20 0.36
SQOR Q9Y6N5 1/20 0.36
DHFR P00374 1/20 0.35
CHRNA7 P36544 1/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8140367 0.86 ACP1 (0.46) ACP1ADORA3F2RL3MAT2ADHODH
SCHEMBL15483442 0.84 ACP1 (0.44) ACP1ADORA3F2RL3MAT2ADHODH
SCHEMBL13954094 0.83 ACP1 (0.44) ACP1ADORA3F2RL3MAT2ADHODH
SCHEMBL13924286 0.82 APP (0.40) ACP1TLR9TLR7PTGDRAPP
SCHEMBL12335705 0.74 ACP1 (0.44) ACP1TLR9TLR7PTGDRAPP
SCHEMBL8273105 0.74 SYK (0.50) ACP1APPKDM4ENPC1RAB9A
SCHEMBL8186120 0.73 ACP1 (0.45) ACP1ADORA3F2RL3MAT2ADHODH
SCHEMBL8191159 0.73 DHODH (0.46) ACP1ADORA3F2RL3MAT2ADHODH
SCHEMBL13444511 0.72 ALDH1A1 (0.47) PTGDRAPPKDM4EMEN1NPC1
SCHEMBL13409339 0.72 APP (0.44) ACP1TLR9TLR7PTGDRAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004094452-A2 MACROCYCLIC ISOQUINOLINE PEPTIDE INHIBITORS OF HEPATITIS C VIRUS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-04 WO disclosed