SCHEMBL12335705

SCHEMBL12335705

COc1ccc2c(OC)nc(-c3cccc(N(C)C)c3)cc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 1/20 0.44
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
VDR P11473 1/20 0.40
CYP2B6 P20813 1/20 0.40
AHR P35869 1/20 0.40
NR1I3 Q14994 1/20 0.40
SQOR Q9Y6N5 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B2 P37059 2/20 0.39
HSD17B1 P14061 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13409378 0.89 MAPT (0.46) ACP1MTNR1AMTNR1BKDM4ESMN1; SMN2
SCHEMBL8353285 0.86 ACP1 (0.43) ACP1MTNR1AMTNR1BKDM4ESMN1; SMN2
SCHEMBL1536561 0.86 ACP1 (0.43) ACP1MTNR1AMTNR1BKDM4ESMN1; SMN2
SCHEMBL1536661 0.86 ACP1 (0.43) ACP1MTNR1AMTNR1BKDM4ESMN1; SMN2
SCHEMBL8300158 0.82 NPC1 (0.59) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL8273117 0.80 MTNR1A (0.42) ACP1MTNR1AMTNR1BKDM4ESMN1; SMN2
SCHEMBL10974850 0.77 ACP1 (0.51) ACP1MTNR1AMTNR1BKDM4EALDH1A1
SCHEMBL8273166 0.76 NPC1 (0.65) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL5068465 0.76 KDM4E (0.45) KDM4EALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL8273091 0.75 RAB9A (0.41) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1505963-B9 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-09-21 EP disclosed
EP-1505963-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-04-20 EP disclosed