SCHEMBL8302676

SCHEMBL8302676

CC(CC#N)c1cccc2cc[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.40
PDPK1 O15530 1/20 0.38
BCHE P06276 3/20 0.37
KEAP1 Q14145 1/20 0.36
NR3C1 P04150 2/20 0.36
PGR P06401 1/20 0.36
NR3C2 P08235 1/20 0.36
AR P10275 1/20 0.36
REN P00797 2/20 0.35
BACE1 P56817 1/20 0.34
BRD4 O60885 1/20 0.33
TAF1 P21675 1/20 0.33
BRPF1 P55201 1/20 0.33
CREBBP Q92793 1/20 0.33
CECR2 Q9BXF3 1/20 0.33
BRD9 Q9H8M2 1/20 0.33
CTSK P43235 2/20 0.32
CTSL P07711 1/20 0.32
CTSS P25774 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3794702 0.80 TSHR (0.44) AHRPDPK1BCHEKEAP1NR3C1
SCHEMBL2611040 0.76 AHR (0.50) AHRPDPK1BCHEKEAP1NR3C1
SCHEMBL14833898 0.74 KEAP1 (0.49) AHRPDPK1BCHEKEAP1NR3C1
SCHEMBL27627249 0.73 ALDH1A1 (0.46)
SCHEMBL29783549 0.73 AHR (0.52) AHRPDPK1BCHEKEAP1NR3C1
SCHEMBL3738852 0.73 AHR (0.52) AHRPDPK1BCHEKEAP1NR3C1
SCHEMBL2260871 0.73 AHR (0.47) AHRPDPK1BCHEKEAP1NR3C1
SCHEMBL1251800 0.70 AHR (0.44) AHRPDPK1BCHEKEAP1NR3C1
SCHEMBL19121929 0.70 BCHE (0.36) AHRBCHE
SCHEMBL2261191 0.69 AHR (0.47) AHRPDPK1KEAP1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469833-B1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY CO ELI (GB) 1999-09-08 EP disclosed
US-5281593-A Pharmaceuticals LILLY INDUSTRIES LIMITED (GB) 1994-01-25 US disclosed
EP-0469833-A1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY INDUSTRIES LIMITED (GB) 1992-02-05 EP disclosed