SCHEMBL8303062

SCHEMBL8303062

Cc1ccc(COC(=O)N2CC/C(=C\C(=O)O)C(F)C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 8/20 0.43
BCL9 O00512 1/20 0.43
CTNNB1 P35222 1/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CYP2C19 P33261 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GRM5 P41594 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300960 0.89 MEN1 (0.44) GRIN2BBCL9CTNNB1MEN1KMT2A
SCHEMBL14500775 0.89 MEN1 (0.44) GRIN2BBCL9CTNNB1MEN1KMT2A
SCHEMBL13712731 0.87 GRIN2B (0.44) GRIN2BBCL9CTNNB1MEN1KMT2A
SCHEMBL13712736 0.87 GRIN2B (0.44) GRIN2BBCL9CTNNB1MEN1KMT2A
SCHEMBL4484409 0.82 GRIN2B (0.47) GRIN2BBCL9CTNNB1MEN1KMT2A
SCHEMBL5149777 0.77 LMNA (0.43) SMN1; SMN2
SCHEMBL5149781 0.77 LMNA (0.43) SMN1; SMN2
SCHEMBL13711175 0.74 GAA (0.37) SMN1; SMN2CYP3A4GRM5
SCHEMBL14099398 0.73 ALDH1A1 (0.44) MEN1KMT2ASMN1; SMN2
SCHEMBL19753633 0.73 GRIN2B (0.54) GRIN2BBCL9CTNNB1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004108705-A1 3-FLUORO-PIPERIDINES AS NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2004-12-16 WO disclosed