SCHEMBL8303575

SCHEMBL8303575

Cc1cc(C(F)(F)F)c(C(N)=O)c(Cl)n1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.65
ALDH1A1 P00352 5/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MAPK1 P28482 1/20 0.49
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAPT P10636 1/20 0.39
HPGD P15428 4/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 3/20 0.38
KDM4E B2RXH2 2/20 0.38
CD38 P28907 1/20 0.37
KCNH2 Q12809 1/20 0.37
TSHR P16473 2/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL565623 0.83 POLB (0.46) POLBALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL27803829 0.79 POLB (1.00) POLBALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL19212155 0.78 POLB (0.76) POLBALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL3749599 0.76 ALDH1A1 (0.44) POLBALDH1A1HPGDLMNAKDM4E
SCHEMBL3753285 0.75 ALDH1A1 (0.44) POLBALDH1A1MAPK1HPGDHSD17B10
SCHEMBL8299880 0.74 HPGD (0.47) POLBALDH1A1SMN1; SMN2MAPK1MAPT
SCHEMBL27764491 0.73 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP2C19HPGDHSD17B10
SCHEMBL27176096 0.72 POLB (0.67) POLBALDH1A1SMN1; SMN2MAPK1CYP1A2
SCHEMBL26852629 0.72 HPGD (0.43) POLBALDH1A1SMN1; SMN2CYP3A4MAPT
SCHEMBL28329012 0.72 KDM4E (0.39) POLBALDH1A1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107382848-A A kind of nicotinamide compounds and its preparation method and application 河北蓝泰化工科技有限公司 2017-11-24 CN disclosed
EP-0429987-B1 5,11-Dihydro-6H-dipyrido[3,2-b:2',3'-e] [1,4]diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMA (US) 1999-03-17 EP disclosed
US-5620974-A ENZYME INHIBITOR, TREATS ACQUIRED IMMUNE DEFICIENCY SYNDROME(AIDS) BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1997-04-15 US disclosed
US-5366972-A 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1994-11-22 US disclosed
EP-0429987-A2 5,11-Dihydro-6H-dipyrido[3,2-b:2',3'-e] [1,4]diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1991-06-05 EP disclosed