SCHEMBL8303898

SCHEMBL8303898

CCOc1ccc(CNC(=O)c2cc(-c3ccccn3)nc3ccc(S(=O)(=O)N4CCOCC4)cc23)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.67
XBP1 P17861 1/20 0.67
MAPT P10636 4/20 0.61
POLB P06746 2/20 0.61
CNR1 P21554 1/20 0.61
ATM Q13315 1/20 0.61
KMT2A Q03164 4/20 0.60
MEN1 O00255 3/20 0.57
RXFP1 Q9HBX9 2/20 0.57
KDM4E B2RXH2 5/20 0.56
HTT P42858 2/20 0.56
APOBEC3G Q9HC16 1/20 0.56
HCRTR1 O43613 1/20 0.56
PPARG P37231 1/20 0.56
NCOA2 Q15596 1/20 0.56
NCOA1 Q15788 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
NCOA3 Q9Y6Q9 1/20 0.56
LMNA P02545 2/20 0.54
TP53 P04637 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308787 0.92 ALDH1A1 (0.79) ALDH1A1XBP1MAPTPOLBCNR1
SCHEMBL8304108 0.83 TSHR (0.66) ALDH1A1XBP1MAPTPOLBCNR1
SCHEMBL8304199 0.83 ALDH1A1 (0.70) ALDH1A1XBP1MAPTPOLBCNR1
SCHEMBL8311922 0.80 HTT (0.65) ALDH1A1XBP1MAPTPOLBCNR1
SCHEMBL8311190 0.79 ALDH1A1 (0.61) ALDH1A1XBP1MAPTPOLBCNR1
SCHEMBL8310878 0.79 ALDH1A1 (0.66) ALDH1A1XBP1MAPTPOLBCNR1
SCHEMBL8308784 0.79 KMT2A (0.67) ALDH1A1XBP1MAPTPOLBCNR1
SCHEMBL8308627 0.78 KMT2A (0.73) ALDH1A1XBP1MAPTPOLBCNR1
SCHEMBL8309338 0.78 ALDH1A1 (0.61) ALDH1A1XBP1MAPTPOLBCNR1
SCHEMBL8311688 0.76 ALDH1A1 (0.65) ALDH1A1XBP1MAPTPOLBCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed