SCHEMBL8308627

SCHEMBL8308627

CC1CCN(CCCNC(=O)c2cc(-c3ccccn3)nc3ccc(S(=O)(=O)N4CCOCC4)cc23)CC1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.73
HTT P42858 2/20 0.68
ALDH1A1 P00352 5/20 0.60
MAPT P10636 2/20 0.60
CNR1 P21554 1/20 0.60
LMNA P02545 3/20 0.58
THRB P10828 1/20 0.58
RXFP1 Q9HBX9 2/20 0.58
POLB P06746 2/20 0.58
ATM Q13315 1/20 0.58
MEN1 O00255 1/20 0.58
XBP1 P17861 1/20 0.55
KCNH2 Q12809 1/20 0.54
KDM4E B2RXH2 2/20 0.53
APOBEC3G Q9HC16 1/20 0.53
CYP2D6 P10635 1/20 0.53
NPSR1 Q6W5P4 1/20 0.52
TSHR P16473 1/20 0.52
BACE1 P56817 1/20 0.52
USP2 O75604 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308784 0.86 KMT2A (0.67) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8308787 0.82 ALDH1A1 (0.79) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8311190 0.82 ALDH1A1 (0.61) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8308067 0.81 KMT2A (0.78) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8311922 0.81 HTT (0.65) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8303840 0.80 KMT2A (0.80) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8304199 0.80 ALDH1A1 (0.70) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8311188 0.80 KMT2A (0.74) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8309338 0.80 ALDH1A1 (0.61) KMT2AHTTALDH1A1MAPTCNR1
SCHEMBL8304108 0.79 TSHR (0.66) KMT2AHTTALDH1A1MAPTCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed