SCHEMBL8303911

SCHEMBL8303911

NC(=O)c1ccc(N2CCCN(CCC3OCCc4ccccc43)CC2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.68
HTR2A P28223 7/20 0.68
DRD4 P21917 6/20 0.68
HTR1A P08908 6/20 0.68
ADRA2A P08913 1/20 0.68
ADRA2B P18089 1/20 0.68
ADRA2C P18825 1/20 0.68
DRD1 P21728 1/20 0.68
ADRA1D P25100 1/20 0.68
ADRA1A P35348 1/20 0.68
ADRA1B P35368 1/20 0.68
DRD3 P35462 1/20 0.68
HTR2B P41595 1/20 0.68
CA12 O43570 1/20 0.68
CA1 P00915 1/20 0.68
CA2 P00918 1/20 0.68
CA4 P22748 1/20 0.68
CA6 P23280 1/20 0.68
CA5A P35218 1/20 0.68
CA7 P43166 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7404186 1.00 DRD2 (0.68) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL5698979 0.96 DRD2 (0.73) DRD2HTR2ADRD4HTR1AADRA2A
Hydrochloric Acid SCHEMBL8178893 0.95 DRD2 (0.72) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL7395270 0.95 DRD2 (0.67) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL7400213 0.90 DRD2 (0.64) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL7395787 0.87 DRD2 (0.72) DRD2HTR2ADRD4HTR1AADRA2A
Hydrochloric Acid SCHEMBL7394797 0.86 DRD2 (0.70) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL7399904 0.85 DRD2 (0.92) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL8551188 0.84 HTR1D (0.78) DRD2HTR2ADRD4HTR1AADRA2A
SCHEMBL7398463 0.83 DRD2 (0.79) DRD2HTR2ADRD4HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737189-B1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS UPJOHN CO (US) 1999-07-28 EP claimed