SCHEMBL8304205

SCHEMBL8304205

C[C@@H]1CCN[C@@H](C(=O)NOCc2ccccc2)C1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.43
RAB9A P51151 7/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
CTSC P53634 1/20 0.43
EPHX2 P34913 2/20 0.43
MASP2 O00187 1/20 0.43
TSHR P16473 1/20 0.40
CPB1 P15086 1/20 0.40
SLC6A2 P23975 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304207 1.00 NPC1 (0.43) NPC1RAB9AHTR2CHTR2BCTSC
Trifluoroacetic Acid SCHEMBL9251606 0.93 CTSC (0.41) NPC1RAB9AHTR2CHTR2BCTSC
Trifluoroacetic Acid SCHEMBL3553696 0.81 HTR2C (0.46) NPC1RAB9AHTR2CHTR2BCTSC
Trifluoroacetic Acid SCHEMBL3553698 0.81 HTR2C (0.46) NPC1RAB9AHTR2CHTR2BCTSC
Hydrochloric Acid SCHEMBL3545786 0.81 HTR2C (0.60) NPC1RAB9AHTR2CHTR2BCTSC
Hydrochloric Acid SCHEMBL3545785 0.81 HTR2C (0.60) NPC1RAB9AHTR2CHTR2BCTSC
SCHEMBL1576471 0.81 TSHR (0.57) HTR2CHTR2BTSHRCPB1
SCHEMBL7996223 0.81 TSHR (0.57) HTR2CHTR2BTSHRCPB1
SCHEMBL7994521 0.81 TSHR (0.57) HTR2CHTR2BTSHRCPB1
SCHEMBL23491956 0.80 MASP2 (0.53) HTR2CHTR2BCTSCMASP2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0614986-B1 Enzymatic racemate cleavage of 2-pipéridine alkylcarboxylates SYNTHELABO (FR) 1999-07-21 EP disclosed
EP-0565396-B1 1-[2-(arylsulfonylamino)-1-oxoethyl]piperidine derivatives, their preparation and use in therapy SYNTHELABO (FR) 1998-01-07 EP disclosed
EP-0614986-A1 Enzymatic racemate cleavage of 2-pipéridine alkylcarboxylates and their use as synthesis intermediates SYNTHELABO (FR) 1994-09-14 EP disclosed
EP-0565396-A1 1-(2-arylsulfonylamino)-1-oxoethyl)-piperidine derivatives, their preparation and use in therapy SYNTHELABO (FR) 1993-10-13 EP disclosed