SCHEMBL8304703

SCHEMBL8304703

CCOC(=O)c1ccc(CSC2NC(=O)C2Br)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
ESR1 P03372 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
ESR2 Q92731 1/20 0.43
CA14 Q9ULX7 1/20 0.43
HTT P42858 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
TSHR P16473 1/20 0.43
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAOA P21397 1/20 0.42
KMT2A Q03164 2/20 0.41
MAPT P10636 5/20 0.40
HPGD P15428 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301620 0.77 CA12 (0.45) CA12CA1CA2ESR1CA7
SCHEMBL128190 0.72 CA1 (0.70) CA12CA1CA2ESR1CA7
SCHEMBL27729402 0.72 CA1 (0.59) CA12CA1CA2ESR1CA7
SCHEMBL27499196 0.70 LMNA (0.61) CA12CA1CA2ESR1CA7
SCHEMBL8302756 0.69 LMNA (0.59) CA12CA1CA2ESR1CA7
SCHEMBL87450 0.69 CA1 (0.83) CA12CA1CA2ESR1CA7
SCHEMBL10943131 0.68 CA1 (0.63) CA12CA1CA2ESR1CA7
SCHEMBL15672816 0.68 CA1 (0.63) CA12CA1CA2ESR1CA7
SCHEMBL245250 0.68 CA1 (0.63) CA12CA1CA2ESR1CA7
SCHEMBL1995591 0.68 CA1 (0.68) CA12CA1CA2ESR1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915843-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSES SMITHKLINE BEECHAM PLC (GB) 1999-05-19 EP disclosed
WO-1997041098-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-11-06 WO disclosed