SCHEMBL8304819

SCHEMBL8304819

Cc1ccc(-c2ccccc2C(F)(F)F)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.50
CCR5 P51681 1/20 0.50
CCR8 P51685 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HSD11B1 P28845 6/20 0.49
CYP3A4 P08684 3/20 0.48
CYP1A2 P05177 3/20 0.48
PDE10A Q9Y233 1/20 0.46
CYP2C19 P33261 3/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2D6 P10635 1/20 0.44
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
KMO O15229 2/20 0.43
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
TRPA1 O75762 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.42
TRPV1 Q8NER1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2406803 0.79 ALOX5AP (0.48) HSD11B1CYP3A4CYP1A2CYP2C19ALDH1A1
SCHEMBL905109 0.79 CYP3A4 (0.55) HSD11B1CYP3A4CYP1A2CYP2C19ALDH1A1
SCHEMBL15060623 0.79 CYP3A4 (0.44) HSD11B1CYP3A4CYP1A2CYP2C19ALDH1A1
SCHEMBL25619166 0.77 CCR1 (0.47) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL12320877 0.77 CYP11B1 (0.56) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL8227859 0.76 CCR1 (0.60) CCR1CCR5CCR8HDAC6CYP3A4
SCHEMBL25303596 0.76 KMO (0.47) HSD11B1CYP3A4CYP1A2CYP2C19ALDH1A1
SCHEMBL8305847 0.76 KMO (0.43) CYP3A4CYP1A2CYP2C19ALDH1A1CYP2D6
SCHEMBL5963839 0.76 KMO (0.43) HSD11B1CYP3A4CYP1A2CYP2C19ALDH1A1
SCHEMBL13017148 0.75 CYP3A4 (0.42) HSD11B1CYP3A4CYP1A2CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023008644-A1 ORGANIC COMPOUND, AND ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAME (주)피엔에이치테크 2023-02-02 WO disclosed
US-5872136-A Arylheteroaryl inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 1999-02-16 US disclosed
EP-0891361-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP disclosed
WO-1997036901-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO disclosed