SCHEMBL905109

SCHEMBL905109

CNc1ccc(-c2ccccc2C(F)(F)F)nc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.55
CYP1A2 P05177 9/20 0.55
CYP2C19 P33261 10/20 0.51
CYP2D6 P10635 7/20 0.51
ALOX15 P16050 4/20 0.51
HSD17B10 Q99714 4/20 0.51
ALDH1A1 P00352 3/20 0.51
MAPK1 P28482 2/20 0.51
PTPN1 P18031 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
USP2 O75604 2/20 0.46
ACP1 P24666 1/20 0.44
TDP1 Q9NUW8 2/20 0.43
RECQL P46063 1/20 0.43
VCP P55072 1/20 0.42
ATR Q13535 1/20 0.41
HSD11B1 P28845 1/20 0.41
SLC22A12 Q96S37 1/20 0.41
TSHR P16473 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304819 0.79 CCR1 (0.50) CYP3A4CYP1A2CYP2C19CYP2D6ALOX15
SCHEMBL26739772 0.79 DHODH (0.51) ALDH1A1MEN1KMT2A
SCHEMBL5964023 0.78 CYP3A4 (0.48) CYP3A4CYP1A2CYP2C19CYP2D6ALOX15
SCHEMBL26739769 0.77 CYP1A2 (0.50) CYP3A4CYP1A2CYP2C19CYP2D6ALOX15
SCHEMBL2406803 0.76 ALOX5AP (0.48) CYP3A4CYP1A2CYP2C19CYP2D6ALOX15
SCHEMBL15060623 0.75 CYP3A4 (0.44) CYP3A4CYP1A2CYP2C19CYP2D6ALOX15
SCHEMBL5964127 0.75 KIF11 (0.53) CYP3A4CYP1A2CYP2C19CYP2D6ALOX15
SCHEMBL905134 0.74 CYP1A2 (0.51) CYP3A4CYP1A2CYP2C19CYP2D6ALOX15
SCHEMBL3152503 0.73 CCR1 (0.46) CYP3A4ALOX15HSD17B10ALDH1A1PTPN1
SCHEMBL5964032 0.73 OXTR (0.48) CYP3A4CYP1A2MAPK1KMT2AATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012043891-A1 AGENT FOR TREATMENT OF EYE DISEASES ダイトーケミックス株式会社 (JP) 2012-04-05 WO disclosed
WO-2012014994-A1 NAPHTHALENE DERIVATIVE ダイトーケミックス株式会社 (JP) 2012-02-02 WO disclosed