SCHEMBL8305007

SCHEMBL8305007

CCCCCCCCC1CCc2cc(-c3ccc(O)cc3)nc(F)c2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
CYP2C8 P10632 2/20 0.39
S1PR3 Q99500 2/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
STAT3 P40763 1/20 0.36
RAB9A P51151 1/20 0.36
ATM Q13315 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
S1PR1 P21453 6/20 0.34
SGPL1 O95470 2/20 0.34
S1PR4 O95977 1/20 0.33
S1PR5 Q9H228 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
ESR2 Q92731 2/20 0.32
ESRRB O95718 1/20 0.32
ESR1 P03372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305593 0.87 XDH (0.40) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL8445620 0.79 ESR2 (0.34) ESR2ESRRBESR1ESRRADRD2
SCHEMBL8296050 0.77 NPC1 (0.34) NPC1MAPTSTAT3RAB9AATM
SCHEMBL8302527 0.77 NPC1 (0.34) NPC1MAPTSTAT3RAB9AATM
SCHEMBL7669115 0.73 CYP3A4 (0.39) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL11188070 0.70 S1PR1 (0.41) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL11185833 0.70 S1PR1 (0.41) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL11185861 0.70 S1PR1 (0.41) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL11179113 0.70 S1PR1 (0.41) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9
SCHEMBL11187996 0.70 S1PR1 (0.41) CYP3A4CYP2C8S1PR3CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824520-B1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AG (DE) 1999-10-06 EP disclosed
US-5942618-A 3,7-DISUBSTITUTED 1-FLUORO-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES HAVING EXCELLENT LIGHT, CHEMICAL AND THERMAL STABILITY; COLORLESS IN PURE STATE; USE IN SWITCHING AND/OR DISPLAY DEVICE HOECHST AKTIENGESELLSCHAFT (DE) 1999-08-24 US disclosed
EP-0824520-A1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-25 EP disclosed
WO-1996035675-A1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AKTIENGESELLSCHAFT (DE) 1996-11-14 WO disclosed