SCHEMBL8305451

SCHEMBL8305451

COc1cc2ncnc(Nc3ccc(OCc4ccc(C(N)=O)cc4)c(C)c3)c2cc1OC

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.63
ERBB2 P04626 2/20 0.63
CLK1 P49759 1/20 0.61
ABCG2 Q9UNQ0 1/20 0.61
LCK P06239 1/20 0.60
KDR P35968 15/20 0.60
RET P07949 3/20 0.58
KIF5B P33176 2/20 0.58
GAK O14976 1/20 0.56
RIPK2 O43353 1/20 0.56
STK10 O94804 1/20 0.56
FLT3 P36888 1/20 0.56
JAK3 P52333 1/20 0.56
AAK1 Q2M2I8 1/20 0.56
Q6ZSR9 Q6ZSR9 1/20 0.56
SLK Q9H2G2 1/20 0.56
IRAK4 Q9NWZ3 1/20 0.56
RPS6KA6 Q9UK32 1/20 0.56
ALK Q9UM73 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5569469 0.86 KDR (0.72) EGFRCLK1ABCG2LCKKDR
SCHEMBL8308795 0.84 KDR (0.74) EGFRERBB2CLK1ABCG2LCK
Hydrochloric Acid SCHEMBL8809576 0.84 EGFR (0.76) EGFRERBB2CLK1ABCG2LCK
SCHEMBL8309890 0.83 EGFR (0.65) EGFRERBB2CLK1ABCG2LCK
SCHEMBL8617925 0.80 MAPK8 (0.46) EGFRKDR
SCHEMBL13889803 0.80 EGFR (0.66) EGFRERBB2CLK1ABCG2LCK
SCHEMBL8307447 0.79 KDR (0.76) EGFRERBB2CLK1ABCG2LCK
SCHEMBL5831668 0.79 ERBB2 (0.75) EGFRERBB2CLK1ABCG2LCK
SCHEMBL5569012 0.79 EGFR (0.72) EGFRERBB2CLK1ABCG2LCK
Hydrochloric Acid SCHEMBL4463390 0.78 ERBB2 (0.73) EGFRERBB2CLK1ABCG2LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed
EP-0790986-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1997-08-27 EP disclosed
WO-1996015118-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1996-05-23 WO disclosed