SCHEMBL8309890

SCHEMBL8309890

COc1cc2ncnc(Nc3ccc(OCc4ccc(C#N)cc4)c(C)c3)c2cc1OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.65
ERBB2 P04626 3/20 0.65
ABCG2 Q9UNQ0 2/20 0.63
PIK3CD O00329 1/20 0.63
PIK3CA P42336 1/20 0.63
PIK3CB P42338 1/20 0.63
PIK3CG P48736 1/20 0.63
CLK1 P49759 1/20 0.60
LCK P06239 3/20 0.59
KDR P35968 10/20 0.57
RET P07949 3/20 0.57
KIF5B P33176 2/20 0.57
EPHA2 P29317 4/20 0.56
GAK O14976 2/20 0.55
RIPK2 O43353 1/20 0.55
STK10 O94804 1/20 0.55
FLT3 P36888 1/20 0.55
JAK3 P52333 1/20 0.55
AAK1 Q2M2I8 1/20 0.55
Q6ZSR9 Q6ZSR9 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8809576 0.86 EGFR (0.76) EGFRERBB2ABCG2CLK1LCK
SCHEMBL8308795 0.86 KDR (0.74) EGFRERBB2ABCG2CLK1LCK
SCHEMBL8305451 0.83 EGFR (0.63) EGFRERBB2ABCG2CLK1LCK
SCHEMBL13889803 0.81 EGFR (0.66) EGFRERBB2ABCG2CLK1LCK
Hydrochloric Acid SCHEMBL8808539 0.80 EGFR (0.63) EGFRERBB2ABCG2PIK3CDPIK3CA
SCHEMBL8307447 0.80 KDR (0.76) EGFRERBB2ABCG2CLK1LCK
SCHEMBL8614554 0.80 CSF1R (0.47) ABCG2FLT3
SCHEMBL7449821 0.79 KDR (0.72) EGFRKDRRETKIF5B
SCHEMBL1387156 0.79 EGFR (0.75) EGFRERBB2ABCG2CLK1LCK
SCHEMBL8306859 0.79 EGFR (1.00) EGFRERBB2ABCG2CLK1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed
EP-0790986-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1997-08-27 EP disclosed
WO-1996015118-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1996-05-23 WO disclosed