SCHEMBL8306147

SCHEMBL8306147

Cc1cccnc1[C@H]1CCC[C@@H](c2ncccc2C)N1Cc1ccc(CNCC(=O)O)cc1CO

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 4/20 0.34
S1PR1 P21453 2/20 0.34
S1PR5 Q9H228 1/20 0.33
HTR5A P47898 1/20 0.33
ALDH1A1 P00352 1/20 0.33
FFAR1 O14842 1/20 0.32
KDM4E B2RXH2 2/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
P2RX7 Q99572 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2475096 0.91 CXCR4 (0.33) CXCR4HTR5AALDH1A1KDM4EPDCD1
SCHEMBL8306155 0.88 CXCR4 (0.35) CXCR4KDM4EP2RX7L3MBTL1
SCHEMBL2474177 0.87 CXCR4 (0.35) CXCR4KDM4EP2RX7
SCHEMBL2473633 0.86 PTGES (0.40) CXCR4KDM4EP2RX7
SCHEMBL11983350 0.86 MAPT (0.36) CXCR4ALDH1A1KDM4EP2RX7
SCHEMBL8301709 0.86 CXCR4 (0.40) CXCR4S1PR1KDM4EL3MBTL1MEN1
SCHEMBL2479491 0.85 SMO (0.35) CXCR4HTR5AKDM4E
SCHEMBL2472333 0.83 CXCR4 (0.38) CXCR4MEN1KMT2A
SCHEMBL2470469 0.83 CXCR4 (0.38) CXCR4MEN1KMT2A
SCHEMBL8302874 0.82 MEN1 (0.45) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090281308-A1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY ANORMED, INC. (CA) 2009-11-12 US disclosed
WO-2004093817-A2 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY ANORMED INC. (CA) 2004-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090281308-A1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY CXCR4, CXCR1, CCR5 CXCR4 1/4885S1PR1 144/4885S1PR5 189/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.