SCHEMBL8306308

SCHEMBL8306308

[O]CCCNCCN1CCOCC1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PAOX Q6QHF9 1/20 0.51
KDM1A O60341 3/20 0.48
ACE2 Q9BYF1 1/20 0.45
HPGD P15428 1/20 0.44
DUSP3 P51452 1/20 0.44
KEAP1 Q14145 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GAA P10253 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
ALDH1A1 P00352 1/20 0.43
RAB9A P51151 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
LMNA P02545 2/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3523671 0.88 KDM1A (0.46) PAOXKDM1AACE2HPGDDUSP3
SCHEMBL4401738 0.85 CA12 (0.53) PAOXKDM1AACE2HPGDDUSP3
SCHEMBL3522928 0.85 PAOX (0.59) PAOXKDM1AHPGDDUSP3KEAP1
SCHEMBL8310197 0.82 ACE2 (0.50) KDM1AACE2SMN1; SMN2CA12CA1
SCHEMBL721355 0.81 PAOX (0.64) PAOXKDM1AHPGDDUSP3KEAP1
SCHEMBL8310938 0.81 KEAP1 (0.64) PAOXKDM1AACE2HPGDDUSP3
SCHEMBL8310934 0.81 KDM1A (0.48) PAOXKDM1AACE2HPGDDUSP3
SCHEMBL29235706 0.81 KDM1A (0.48) PAOXKDM1AACE2HPGDDUSP3
SCHEMBL13912969 0.81 PAOX (0.51) PAOXKDM1AACE2HPGDDUSP3
SCHEMBL8306310 0.81 ALDH1A1 (0.53) PAOXKDM1AACE2HPGDDUSP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed
US-5821246-A USEFUL AS TYROSINE KINASE INHIBITORS AND FOR THE TREATMENT OF PROLIFERATIVE DISEASES SUCH AS CANCER ZENECA LIMITED (GB) 1998-10-13 US disclosed
EP-0790986-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1997-08-27 EP disclosed
WO-1996015118-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1996-05-23 WO disclosed