SCHEMBL8306799

SCHEMBL8306799

COC(=O)c1cc(OCC#N)c2[nH]ccc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.39
CYP3A4 P08684 1/20 0.36
BCHE P06276 3/20 0.36
POLB P06746 2/20 0.36
ALOX15 P16050 2/20 0.36
HTT P42858 2/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36
TUBB8 Q3ZCM7 1/20 0.36
TUBA3E Q6PEY2 1/20 0.36
TUBA1A Q71U36 1/20 0.36
TUBA1C Q9BQE3 1/20 0.36
TUBB6 Q9BUF5 1/20 0.36
TUBB2B Q9BVA1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18031228 0.82 CYP3A4 (0.50) CDK8CYP3A4BCHEPOLBTUBB4A
SCHEMBL18033368 0.81 NPC1 (0.44) CDK8BCHEALDH1A1MAPTKDM4E
SCHEMBL18009394 0.79 HPGD (0.55) CYP3A4LMNAMAPTSMN1; SMN2MEN1
SCHEMBL18031516 0.78 P2RX7 (0.43) CDK8CYP3A4BCHEPOLBALOX15
SCHEMBL15971072 0.78 POLB (0.41) CDK8CYP3A4POLBALOX15TUBB4A
SCHEMBL18033213 0.75 POLB (0.39) CDK8CYP3A4BCHEPOLBHTT
SCHEMBL143239 0.74 CDK8 (0.44) CDK8POLBALOX15HTTALDH1A1
SCHEMBL18031517 0.74 KDM4E (0.53) CDK8POLBALOX15HTTALDH1A1
SCHEMBL8301795 0.73 PIM3 (0.43) ALDH1A1LMNAMAPTSMN1; SMN2MEN1
SCHEMBL15595537 0.73 MAPT (0.59) CYP3A4ALDH1A1LMNAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469833-B1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY CO ELI (GB) 1999-09-08 EP disclosed
US-5281593-A Pharmaceuticals LILLY INDUSTRIES LIMITED (GB) 1994-01-25 US disclosed
EP-0469833-A1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY INDUSTRIES LIMITED (GB) 1992-02-05 EP disclosed