SCHEMBL8306870

SCHEMBL8306870

COC(=O)CCc1c(C(=O)c2ccc(Cl)cc2)oc2cc(NC(=O)CC(=O)OC)ccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
L3MBTL1 Q9Y468 4/20 0.39
NPSR1 Q6W5P4 3/20 0.39
KDM4E B2RXH2 4/20 0.39
HPGD P15428 4/20 0.39
MAPT P10636 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
ALOX12 P18054 1/20 0.39
HTT P42858 1/20 0.39
THRB P10828 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
CA12 O43570 2/20 0.38
CA9 Q16790 2/20 0.38
POLB P06746 2/20 0.37
RAD52 P43351 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9070589 0.91 CA12 (0.43) ALDH1A1L3MBTL1NPSR1KDM4EHPGD
SCHEMBL8841213 0.91 KDM4E (0.41) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL8326230 0.86 CYP19A1 (0.44) ALDH1A1L3MBTL1NPSR1KDM4EHPGD
SCHEMBL679245 0.85 ALDH1A1 (0.46) ALDH1A1L3MBTL1NPSR1KDM4EHPGD
SCHEMBL27445439 0.84 SMN1; SMN2 (0.43) ALDH1A1L3MBTL1NPSR1KDM4EHPGD
SCHEMBL9070592 0.83 KDM4E (0.45) ALDH1A1L3MBTL1NPSR1KDM4EHPGD
SCHEMBL8554638 0.82 ALDH1A1 (0.40) ALDH1A1L3MBTL1NPSR1KDM4EHPGD
SCHEMBL8557494 0.82 ALDH1A1 (0.39) ALDH1A1L3MBTL1NPSR1KDM4EHPGD
SCHEMBL8307013 0.81 ALDH1A1 (0.45) ALDH1A1L3MBTL1NPSR1KDM4EHPGD
SCHEMBL27445438 0.78 SMN1; SMN2 (0.46) ALDH1A1L3MBTL1NPSR1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0685475-B1 Amino-benzofuryl-and thienyl-derivatives BAYER AG (DE) 1999-01-13 EP disclosed
EP-0685474-B1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1998-09-16 EP disclosed
US-5622989-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
US-5565488-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-10-15 US disclosed
EP-0685475-A1 Amino-benzofuryl-and thienyl-derivatives BAYER AG (DE) 1995-12-06 EP disclosed
EP-0685474-A1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1995-12-06 EP disclosed