SCHEMBL8307208

SCHEMBL8307208

N=C(N)c1cccc(CNc2ncnc3cc(C(=O)N4CCCC4)ccc23)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 5/20 0.48
PRSS1 P07477 2/20 0.48
AURKA O14965 5/20 0.47
RPS6KB1 P23443 5/20 0.47
AURKB Q96GD4 5/20 0.47
PDE5A O76074 1/20 0.47
MAPK10 P53779 4/20 0.46
MAPK8 P45983 3/20 0.46
NPC1 O15118 1/20 0.46
LMNA P02545 1/20 0.46
POLB P06746 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.44
CDK1 P06493 1/20 0.44
NTRK1 P04629 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6322361 0.99 AURKA (0.49) F10PRSS1AURKARPS6KB1AURKB
Hydrochloric Acid SCHEMBL6325502 0.99 F10 (0.47) F10PRSS1AURKARPS6KB1AURKB
SCHEMBL6325892 0.98 F10 (0.48) F10PRSS1AURKARPS6KB1AURKB
SCHEMBL6329960 0.92 F10 (0.48) F10PRSS1AURKARPS6KB1AURKB
Hydrochloric Acid SCHEMBL6326766 0.91 F10 (0.48) F10PRSS1AURKARPS6KB1AURKB
SCHEMBL6323988 0.90 CDK1 (0.45) AURKARPS6KB1AURKBPDE5AMAPK10
SCHEMBL6326456 0.89 AURKA (0.41) F10PRSS1AURKARPS6KB1AURKB
SCHEMBL6323907 0.88 CDK1 (0.50) AURKARPS6KB1AURKBPDE5AMAPK10
SCHEMBL6322321 0.86 AURKA (0.42) AURKARPS6KB1AURKBPDE5ANPC1
SCHEMBL6329487 0.86 AURKA (0.43) AURKARPS6KB1AURKBPDE5AMAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080970-A1 NOVEL BICYCLIC AROMATIC COMPOUNDS, THE PRODUCTION AND USE THEREOF IN THE FORM OF DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-09-23 WO disclosed