SCHEMBL8307655

SCHEMBL8307655

COC1C=CC(c2cc(C(F)(F)F)nn2-c2ccc(N)cc2)=CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.54
PTGS1 P23219 10/20 0.46
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
TSHR P16473 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
THPO P40225 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PDPK1 O15530 2/20 0.39
PTGES O14684 1/20 0.38
HDAC3 O15379 1/20 0.38
CA12 O43570 1/20 0.38
PDE5A O76074 1/20 0.38
ABCB11 O95342 1/20 0.38
MT-CO2 P00403 1/20 0.38
CA1 P00915 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14401040 0.74 PTGS2 (0.59) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL8297317 0.73 PTGS2 (0.41) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL8292733 0.70 PTGS2 (1.00) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL7326690 0.69 PTGS2 (0.64) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL14747609 0.68 PTGS2 (0.74) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL5420747 0.68 PTGS2 (0.74) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL14747587 0.68 PTGS2 (0.66) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL3277875 0.68 PTGS1 (0.80) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL14958860 0.67 PDPK1 (0.73) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL2694817 0.67 PTGS2 (0.82) PTGS2PTGS1CYP3A4CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004103286-A2 COMPOSITIONS OF A CYCLOOXYGENASE-2 SELECTIVE INHIBITOR AND A CHOLIMERGIC AGENT PHARMACIA CORPORATION (US) 2004-12-02 WO disclosed