SCHEMBL8307717

SCHEMBL8307717

COc1ccc(-c2cnc(N)c(C(=O)c3ccccc3)n2)cc1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ATR Q13535 15/20 0.69
PRKDC P78527 6/20 0.69
RXFP1 Q9HBX9 1/20 0.51
ATM Q13315 3/20 0.51
NEK2 P51955 1/20 0.51
CDK5 Q00535 1/20 0.51
CDK5R1 Q15078 1/20 0.51
CHEK1 O14757 1/20 0.50
PARP1 P09874 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11907360 0.88 ATR (0.70) ATRPRKDCATMNEK2CHEK1
SCHEMBL5684569 0.87 ATR (0.63) ATRPRKDCATMCDK5CDK5R1
SCHEMBL8306689 0.84 ATR (0.67) ATRPRKDCATMCDK5CDK5R1
SCHEMBL2484387 0.82 ATR (1.00) ATRPRKDCATM
SCHEMBL13912898 0.80 MAPK14 (0.46) ATRPRKDCRXFP1ATMCDK5
SCHEMBL3460862 0.80 ATR (0.72) ATRPRKDCATM
SCHEMBL557954 0.79 ATR (0.72) ATRPRKDCATM
SCHEMBL3462566 0.77 ATR (0.66) ATRPRKDCATM
SCHEMBL14067883 0.77 ATR (0.60) ATRPRKDCATM
SCHEMBL318797 0.76 ATR (0.68) ATRPRKDCATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0914318-A1 PYRAZINES KINGS COLLEGE LONDON (GB) 1999-05-12 EP disclosed
EP-0904272-A1 DIHYDROBENZOFURAN AND RELATED COMPOUNDS USEFUL AS ANTI-INFLAMMATORY AGENTS THE PROCTER & GAMBLE COMPANY (US) 1999-03-31 EP disclosed
WO-1997043267-A1 PYRAZINES KINGS COLLEGE LONDON (GB) 1997-11-20 WO disclosed
WO-1997028155-A1 DIHYDROBENZOFURAN AND RELATED COMPOUNDS USEFUL AS ANTI-INFLAMMATORY AGENTS THE PROCTER & GAMBLE COMPANY (US) 1997-08-07 WO disclosed