SCHEMBL8307974

SCHEMBL8307974

FC1(F)CCC(Nc2ncnc3cnc(NCCN4CCOCC4)cc23)CC1

nearest known ligand 0.80

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.58
IRAK4 Q9NWZ3 2/20 0.52
CYP1A2 P05177 4/20 0.46
CYP3A4 P08684 4/20 0.46
CYP2D6 P10635 4/20 0.46
CLK4 Q9HAZ1 3/20 0.46
HSD17B10 Q99714 3/20 0.46
ALDH1A1 P00352 2/20 0.46
USP2 O75604 1/20 0.46
MAP3K8 P41279 1/20 0.45
LMNA P02545 1/20 0.45
HIF1A Q16665 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312604 0.89 EGFR (0.61) EGFRIRAK4CYP1A2CYP3A4CYP2D6
SCHEMBL8312988 0.78 EGFR (0.57) EGFRCYP1A2CYP3A4CYP2D6CLK4
SCHEMBL4780623 0.78 CYP1A2 (0.59) IRAK4CYP1A2CYP3A4CYP2D6CLK4
SCHEMBL4468260 0.77 EGFR (0.60) EGFRCYP1A2CYP3A4CYP2D6CLK4
SCHEMBL8311954 0.77 CLK1 (0.46) IRAK4CLK4HSD17B10ALDH1A1LMNA
SCHEMBL18359127 0.76 EGFR (0.70) EGFRMAP3K8
SCHEMBL8312573 0.75 EGFR (0.52) EGFR
SCHEMBL6364052 0.73 IRAK4 (0.47) EGFRIRAK4
SCHEMBL18359136 0.72 EGFR (0.73) EGFRCYP1A2CYP3A4CYP2D6CLK4
SCHEMBL6368598 0.71 IRAK4 (0.48) EGFRIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016925-A1 AZAQUINAZOLINE DERIVATIVES PFIZER LIMITED (GB) 2005-02-24 WO disclosed