SCHEMBL8312604

SCHEMBL8312604

c1nc(NC2CCCCC2)c2cc(NCCN3CCOCC3)ncc2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.61
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
CLK4 Q9HAZ1 2/20 0.48
IRAK4 Q9NWZ3 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
USP2 O75604 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MAP3K8 P41279 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8307974 0.89 EGFR (0.58) EGFRCYP1A2CYP3A4CYP2D6CLK4
SCHEMBL4780623 0.88 CYP1A2 (0.59) CYP1A2CYP3A4CYP2D6CLK4IRAK4
SCHEMBL8312573 0.85 EGFR (0.52) EGFRMEN1KMT2A
SCHEMBL8312988 0.82 EGFR (0.57) EGFRCYP1A2CYP3A4CYP2D6CLK4
SCHEMBL6368598 0.82 IRAK4 (0.48) EGFRIRAK4
SCHEMBL8306375 0.80 GRM1 (0.49)
SCHEMBL8312990 0.80 MEN1 (0.44) IRAK4MEN1KMT2A
SCHEMBL4468260 0.79 EGFR (0.60) EGFRCYP1A2CYP3A4CYP2D6CLK4
SCHEMBL8306177 0.78 GRM1 (0.55) EGFR
SCHEMBL18359127 0.77 EGFR (0.70) EGFRMAP3K8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016925-A1 AZAQUINAZOLINE DERIVATIVES PFIZER LIMITED (GB) 2005-02-24 WO disclosed