SCHEMBL8308022

SCHEMBL8308022

CCOC(=O)Cc1cc2cccc(Cl)c2n(Cc2nc3c(F)c(F)ccc3s2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 9/20 0.42
RXFP1 Q9HBX9 1/20 0.37
P2RX7 Q99572 1/20 0.36
AKR1A1 P14550 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
ALDH1A1 P00352 4/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 2/20 0.34
KDM4E B2RXH2 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303795 0.79 AKR1B1 (0.48) AKR1B1RXFP1AKR1A1MEN1KMT2A
SCHEMBL8303442 0.78 AKR1B1 (0.49) AKR1B1RXFP1P2RX7MEN1KMT2A
SCHEMBL8307388 0.75 AKR1B1 (0.56) AKR1B1AKR1A1
SCHEMBL8305325 0.75 AKR1A1 (0.47) AKR1B1AKR1A1
SCHEMBL8304794 0.74 AKR1B1 (0.47) AKR1B1RXFP1AKR1A1MEN1KMT2A
SCHEMBL8303689 0.74 KDM4E (0.40) AKR1B1RXFP1MEN1KMT2AALDH1A1
SCHEMBL8307232 0.73 AKR1B1 (0.60) AKR1B1AKR1A1
SCHEMBL8304134 0.72 AKR1B1 (0.54) AKR1B1AKR1A1
SCHEMBL8307246 0.72 AKR1B1 (0.54) AKR1B1AKR1A1
SCHEMBL8304777 0.71 AKR1B1 (0.45) AKR1B1AKR1A1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0633261-B1 QUINOLINE-3-ACETIC ACID DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF YOSHITOMI PHARMACEUTICAL (JP) 1999-04-21 EP disclosed
US-5543420-A ALDOSE REDUCTASE INHIBITORS; ANTIDIABETIC AGENTS; PREVENTION OF ACCUMULATION OF SORBITOL AND GALACTITOL IN MAMMALIAN TISSUE THE GREEN CROSS CORPORATION (JP) 1996-08-06 US disclosed
EP-0633261-A1 QUINOLINE-3-ACETIC ACID DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF THE GREEN CROSS CORPORATION (JP) 1995-01-11 EP disclosed