SCHEMBL8308397

SCHEMBL8308397

Nc1c(Cl)cc(-c2nn(C3CCN(CCCC(F)(F)F)CC3)c(=O)o2)c2c1OCCO2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 15/20 0.49
HTR2C P28335 3/20 0.39
HTR3A P46098 3/20 0.39
HTR3E A5X5Y0 2/20 0.39
HTR3B O95264 2/20 0.39
HTR3D Q70Z44 2/20 0.39
HTR3C Q8WXA8 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
ADRA2A P08913 2/20 0.39
HTR2A P28223 2/20 0.39
ADRA1A P35348 2/20 0.39
LMNA P02545 1/20 0.39
THRB P10828 1/20 0.39
ADRA2C P18825 1/20 0.39
HTR1D P28221 1/20 0.39
HRH1 P35367 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306432 0.89 HTR4 (0.53) HTR4HTR2CHTR3AHTR3EHTR3B
Hydrochloric Acid SCHEMBL8364693 0.88 HTR4 (0.52) HTR4HTR2CHTR3AHTR3EHTR3B
SCHEMBL8307419 0.85 HTR4 (0.36) HTR4HTR2CHTR3AADRA2AHTR2A
SCHEMBL8303718 0.83 HTR4 (0.52) HTR4
SCHEMBL8309195 0.83 HTR4 (0.42) HTR4HTR2CHTR2AHTR2BNPSR1
Capeserod SCHEMBL4707724 0.83 HTR4 (0.45) HTR4HTR2CHTR3AHTR3EHTR3B
Bromide SCHEMBL8369649 0.82 HTR4 (0.51) HTR4
Capeserod SCHEMBL399091 0.82 HTR4 (0.44) HTR4HTR2CHTR3AADRA2AHTR2A
SCHEMBL8364833 0.81 HTR4 (0.46) HTR4HTR2CHTR3AHTR3EHTR3B
SCHEMBL7749161 0.81 HTR4 (0.45) HTR4HTR2CHTR3AHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929089-A ANTISEROTONINE AGENT SYNTHELABO (FR) 1999-07-27 US disclosed
EP-0863897-B1 5-PHENYL-3-(PIPERIDIN-4-YL)-1,3,4-OXADIAZOL-2(3H)-ONE DERIVATIVES FOR USE AS 5-HT4- OR H3-RECEPTOR LIGANDS SYNTHELABO (FR) 1999-06-16 EP disclosed