SCHEMBL8308878

SCHEMBL8308878

O=C(c1ccc(Nc2nccc(-c3ccc(Cl)cc3)n2)cc1)N1CCC(NC2CCCCC2)CC1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.53
IKBKB O14920 12/20 0.49
CHUK O15111 8/20 0.49
IKBKG Q9Y6K9 7/20 0.49
MEN1 O00255 1/20 0.49
RECQL P46063 1/20 0.49
BLM P54132 1/20 0.49
KMT2A Q03164 1/20 0.49
PRKCZ Q05513 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
PIK3CA P42336 2/20 0.49
PIK3CB P42338 2/20 0.49
PIK3CG P48736 2/20 0.49
MTOR P42345 1/20 0.49
SMG1 Q96Q15 1/20 0.49
EPHX2 P34913 1/20 0.48
CDK2 P24941 1/20 0.48
JAK2 O60674 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312581 0.95 CDK1 (0.58) CDK1IKBKBCHUKIKBKGMEN1
SCHEMBL8311072 0.89 DGAT1 (0.49) CDK1IKBKBCHUKIKBKGMEN1
SCHEMBL13590857 0.89 CDK1 (0.54) CDK1IKBKBCHUKIKBKGMEN1
SCHEMBL11924740 0.88 MTOR (0.51) CDK1IKBKBCHUKIKBKGMEN1
SCHEMBL11924733 0.88 MTOR (0.60) IKBKBCHUKIKBKGMEN1RECQL
SCHEMBL14021190 0.88 MTOR (0.60) IKBKBCHUKIKBKGMEN1RECQL
Hydrochloric Acid SCHEMBL4071661 0.88 CDK1 (0.53) CDK1IKBKBCHUKIKBKGMEN1
SCHEMBL8247959 0.88 IKBKB (0.63) IKBKBCHUKIKBKGMEN1RECQL
SCHEMBL8254568 0.88 JAK2 (0.55) IKBKBCHUKIKBKGMEN1RECQL
SCHEMBL14021219 0.87 PIK3CA (0.58) IKBKBCHUKIKBKGPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7442699-B2 Anilinopyrimidine derivatives as IKK inhibitors and compositions and methods related thereto SIGNAL PHARMACEUTICALS, LLC (US) 2008-10-28 US disclosed
US-7442699-B2 Anilinopyrimidine derivatives as IKK inhibitors and compositions and methods related thereto SIGNAL PHARMACEUTICALS, LLC (US) 2008-10-28 US disclosed
US-7429599-B2 Methods for treating or preventing an inflammatory or metabolic condition or inhibiting JNK SIGNAL PHARMACEUTICALS, LLC (US) 2008-09-30 US disclosed
US-7429599-B2 Methods for treating or preventing an inflammatory or metabolic condition or inhibiting JNK SIGNAL PHARMACEUTICALS, LLC (US) 2008-09-30 US disclosed
WO-2004084901-A1 METHODS FOR TREATING OR PREVENTING AN INFLAMMATORY OR METABOLIC CONDITION BY INHIBITING JNK SIGNAL PHARMACEUTICALS, LLC (US) 2004-10-07 WO disclosed