SCHEMBL8309767

SCHEMBL8309767

N#Cc1ccc(Oc2ccc(C(c3ccccc3)(c3ccccc3)c3ncc[nH]3)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.46
CHEK2 O96017 1/20 0.39
MAOB P27338 1/20 0.39
TTBK1 Q5TCY1 1/20 0.39
TTBK2 Q6IQ55 1/20 0.39
CSNK1A1 P48729 1/20 0.38
CSNK1D P48730 1/20 0.38
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
TNK2 Q07912 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 7/20 0.36
KCNH2 Q12809 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN9A Q15858 1/20 0.36
PARP15 Q460N3 1/20 0.35
PARP10 Q53GL7 1/20 0.35
PARP2 Q9UGN5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11863909 0.89 KIF11 (0.39) CYP19A1MAOBMEN1KIF11CYP11B1
SCHEMBL8306983 0.85 TAAR1 (0.40) CYP19A1MAOBGRIN1GRIN2BMEN1
SCHEMBL8099648 0.83 CYP19A1 (0.36) CYP19A1TTBK1TTBK2LMNASMN1; SMN2
Trityl Imidazole SCHEMBL1572623 0.78 MTOR (0.45) CYP19A1LMNASMN1; SMN2MEN1CYP11B1
SCHEMBL8309765 0.75 LMNA (0.40) CYP19A1CHEK2MAOBCSNK1A1CSNK1D
SCHEMBL11089506 0.75 MTOR (0.45) CYP19A1LMNASMN1; SMN2MEN1CYP11B1
SCHEMBL9669719 0.75 TAAR1 (0.36) CYP19A1LMNASMN1; SMN2
SCHEMBL1484199 0.73 CYP19A1 (0.41) CYP19A1KIF11
SCHEMBL5738213 0.73 NISCH (0.43) CYP19A1LMNASMN1; SMN2MEN1KIF11
SCHEMBL3827055 0.73 CYP19A1 (0.41) CYP19A1CSNK1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891333-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP disclosed
WO-1997036875-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO disclosed