SCHEMBL8309844

SCHEMBL8309844

CC(=O)CCOC(=O)/N=C(\N)c1ccc(O)c(CNc2ncnc3cc(C(=O)N4CCCC4)c(C)cc23)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.34
PDE5A O76074 3/20 0.34
AURKA O14965 4/20 0.32
AURKB Q96GD4 2/20 0.32
ALDH1A1 P00352 3/20 0.32
HPGD P15428 2/20 0.32
HTT P42858 2/20 0.32
RPS6KB1 P23443 3/20 0.31
EGFR P00533 3/20 0.30
USP2 O75604 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
CYP2C19 P33261 1/20 0.30
HSD17B10 Q99714 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
LMNA P02545 1/20 0.30
CNR1 P21554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308730 0.92 PDE5A (0.36) CDK1PDE5AAURKAAURKBALDH1A1
SCHEMBL8312292 0.85 CDK1 (0.36) CDK1PDE5AAURKAAURKBALDH1A1
SCHEMBL8308640 0.84 CDK1 (0.37) CDK1PDE5AALDH1A1HPGDEGFR
SCHEMBL2991625 0.83 F10 (0.41) CDK1PDE5AAURKAAURKBALDH1A1
SCHEMBL8312245 0.81 HPGD (0.36) CDK1PDE5AALDH1A1HPGDHTT
SCHEMBL3000544 0.79 CDK1 (0.40) CDK1PDE5AALDH1A1HPGDHTT
SCHEMBL2995881 0.79 PDE5A (0.36) CDK1PDE5AALDH1A1HPGDHTT
SCHEMBL8311630 0.78 CDK1 (0.42) CDK1PDE5AAURKAAURKBALDH1A1
SCHEMBL8312247 0.77 CDK1 (0.39) CDK1PDE5AAURKAAURKBALDH1A1
SCHEMBL6327115 0.75 CDK1 (0.37) CDK1PDE5AAURKAAURKBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080970-A1 NOVEL BICYCLIC AROMATIC COMPOUNDS, THE PRODUCTION AND USE THEREOF IN THE FORM OF DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-09-23 WO disclosed