SCHEMBL8309926

SCHEMBL8309926

Nc1ccc(C(=O)c2cccnc2)c(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.50
ALDH1A1 P00352 3/20 0.50
NPC1 O15118 3/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
MKNK1 Q9BUB5 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
JAK2 O60674 1/20 0.49
TYK2 P29597 1/20 0.49
F7 P08709 1/20 0.47
F3 P13726 1/20 0.47
SARM1 Q6SZW1 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.47
SIRT6 Q8N6T7 1/20 0.47
SIRT1 Q96EB6 1/20 0.47
SIRT3 Q9NTG7 1/20 0.47
SIRT5 Q9NXA8 1/20 0.47
SIRT4 Q9Y6E7 1/20 0.47
KMT2A Q03164 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28077179 0.83 HDAC1 (0.52) ALDH1A1F7F3SARM1SIRT2
SCHEMBL7116217 0.82 MKNK1 (0.49) RAB9AALDH1A1NPC1MKNK1MKNK2
SCHEMBL8309451 0.81 JAK2 (0.61) RAB9AALDH1A1NPC1JAK2TYK2
SCHEMBL5963546 0.81 MAPK13 (0.58) ALDH1A1JAK2TYK2KMT2AMEN1
SCHEMBL7194395 0.80 HSD17B10 (0.58) ALDH1A1NPC1JAK2TYK2KMT2A
SCHEMBL6770549 0.80 HPGD (0.59) RAB9AALDH1A1NPC1F7F3
SCHEMBL7397552 0.79 CCR9 (0.54) RAB9AALDH1A1NPC1NFKB1NFKB2
SCHEMBL28232 0.78 CCR9 (0.58) RAB9AALDH1A1NPC1NFKB1NFKB2
SCHEMBL7183309 0.77 SRD5A2 (0.54) RAB9AALDH1A1JAK2TYK2KMT2A
Chlorobenzene SCHEMBL27529703 0.77 MAPK14 (0.55) RAB9AALDH1A1KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed
US-5821246-A USEFUL AS TYROSINE KINASE INHIBITORS AND FOR THE TREATMENT OF PROLIFERATIVE DISEASES SUCH AS CANCER ZENECA LIMITED (GB) 1998-10-13 US disclosed
EP-0790986-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1997-08-27 EP disclosed
WO-1996015118-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1996-05-23 WO disclosed