SCHEMBL8310019

SCHEMBL8310019

Cc1ccc(N)cc1OCc1nccs1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
HPGD P15428 2/20 0.51
RAB9A P51151 2/20 0.40
MAPT P10636 3/20 0.39
CYP2C19 P33261 1/20 0.39
LMNA P02545 1/20 0.38
SYK P43405 1/20 0.37
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
CASP1 P29466 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
RIPK2 O43353 1/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
YES1 P07947 1/20 0.34
FECH P22830 1/20 0.34
ERBB4 Q15303 1/20 0.34
RIPK3 Q9Y572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310026 0.88 ALDH1A1 (0.42) ALDH1A1HPGDRAB9AMAPTCYP2C19
SCHEMBL2986980 0.79 EGFR (0.44) ALDH1A1HPGDRAB9AMAPTCYP2C19
SCHEMBL25236899 0.76 ALDH1A1 (0.37) ALDH1A1HPGDMAPTCYP2C19LMNA
SCHEMBL6795023 0.74 CYP2C19 (0.48) ALDH1A1RAB9AMAPTCYP2C19GAA
SCHEMBL1188568 0.73 MAPT (0.61) ALDH1A1HPGDRAB9AMAPTKDM4E
SCHEMBL18605599 0.73 CYP3A4 (0.53) ALDH1A1HPGDRAB9ACYP2C19LMNA
SCHEMBL12851558 0.72 KDM4E (0.48) ALDH1A1RAB9AMAPTLMNAKDM4E
SCHEMBL27771618 0.72 ALDH1A1 (0.43) ALDH1A1HPGD
SCHEMBL8307415 0.72 SYK (0.47) ALDH1A1HPGDRAB9AMAPTSYK
SCHEMBL6190711 0.72 SYK (0.69) SYKEGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed
US-5821246-A USEFUL AS TYROSINE KINASE INHIBITORS AND FOR THE TREATMENT OF PROLIFERATIVE DISEASES SUCH AS CANCER ZENECA LIMITED (GB) 1998-10-13 US disclosed
EP-0790986-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1997-08-27 EP disclosed
WO-1996015118-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1996-05-23 WO disclosed