SCHEMBL8310685

SCHEMBL8310685

COC(=O)C1CCCC(N)=N1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 12/20 0.46
NOS2 P35228 12/20 0.46
NOS3 P29474 10/20 0.46
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8308928 0.98 NOS1 (0.44) NOS1NOS2NOS3
SCHEMBL31264948 0.89 CYP2C19 (0.42) NOS1NOS2NOS3CYP2C19KMT2A
Hydrochloric Acid SCHEMBL31264976 0.87 NOS3 (0.44) NOS1NOS2NOS3CYP2C19KMT2A
SCHEMBL31585483 0.82 CHRM2 (0.33)
SCHEMBL9373328 0.77 NOS1 (0.47) NOS1NOS2NOS3CYP2C19
Hydrochloric Acid SCHEMBL8306795 0.76 NOS1 (0.45) NOS1NOS2NOS3
SCHEMBL24664106 0.74 POLB (0.33)
SCHEMBL907524 0.74 POLB (0.33)
SCHEMBL433180 0.74 POLB (0.33)
SCHEMBL18733223 0.72 NOS1 (0.43) NOS1NOS2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630244-B1 MUSCARINIC AGONISTS UNIV TOLEDO (US) 1999-12-01 EP disclosed
US-5403845-A Cognition activators; Alzheimer*s disaease UNIVERSITY OF TOLEDO (US) 1995-04-04 US disclosed
EP-0630244-A1 MUSCARINIC AGONISTS THE UNIVERSITY OF TOLEDO (US) 1994-12-28 EP disclosed
EP-0630244-A4 MUSCARINIC AGONISTS. UNIV TOLEDO (US) 1994-04-07 EP disclosed
WO-1993003726-A1 MUSCARINIC AGONISTS THE UNIVERSITY OF TOLEDO (US) 1993-03-04 WO disclosed
US-5175166-A Cognition activators THE UNIVERSITY OF TOLEDO (US) 1992-12-29 US disclosed