SCHEMBL8311787

SCHEMBL8311787

O=C(O)N1CCC(N(CCC(c2ccccc2)c2ccccc2)Cc2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.55
MEN1 O00255 3/20 0.55
ALDH1A1 P00352 1/20 0.53
CCR5 P51681 10/20 0.46
RAB9A P51151 1/20 0.45
OPRM1 P35372 1/20 0.44
OPRL1 P41146 1/20 0.44
CHRM2 P08172 1/20 0.43
CHRM3 P20309 1/20 0.43
AGTR2 P50052 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978433 0.86 MEN1 (0.53) KMT2AMEN1ALDH1A1CCR5RAB9A
SCHEMBL29243353 0.80 MEN1 (0.50) KMT2AMEN1ALDH1A1CCR5RAB9A
SCHEMBL6978832 0.78 SLC6A2 (0.62)
SCHEMBL28404291 0.75 ALDH1A1 (0.54) KMT2AMEN1ALDH1A1CCR5RAB9A
SCHEMBL16757240 0.74 KMT2A (0.69) KMT2AMEN1ALDH1A1CCR5RAB9A
SCHEMBL785972 0.74 JAK2 (0.54) KMT2AMEN1ALDH1A1OPRM1CHRM2
SCHEMBL16757186 0.73 KMT2A (0.65) KMT2AMEN1ALDH1A1CCR5RAB9A
SCHEMBL20959482 0.73 ALDH1A1 (0.56) KMT2AMEN1ALDH1A1CCR5
SCHEMBL16321987 0.72 KMT2A (0.50) KMT2AMEN1ALDH1A1CCR5
SCHEMBL8311276 0.72 SOS1 (0.58) KMT2AMEN1CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-A1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS Takeda Chemical Industries, Ltd. (JP) 1999-06-23 EP disclosed
WO-1998008842-A1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-05 WO disclosed