SCHEMBL8312588

SCHEMBL8312588

CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CC(F)(F)C1C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.44
CTSL P07711 2/20 0.44
CTSB P07858 1/20 0.44
ELANE P08246 2/20 0.43
HDAC8 Q9BY41 1/20 0.42
PREP P48147 1/20 0.40
CTSS P25774 1/20 0.39
CMA1 P23946 8/20 0.39
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3601920 0.82 HDAC8 (0.47) CTSKCTSLCTSBELANEHDAC8
SCHEMBL5203233 0.75 PIN1 (0.54) CTSKCTSLCTSBELANEHDAC8
SCHEMBL8161374 0.75 CMA1 (0.53) CTSKCTSLCTSBELANECMA1
SCHEMBL8143604 0.75 CMA1 (0.53) CTSKCTSLCTSBELANECMA1
SCHEMBL3611500 0.74 CTSK (0.50) CTSKCTSLCTSBELANEHDAC8
SCHEMBL22169449 0.74 CTSK (0.50) CTSKCTSLCTSBELANEHDAC8
SCHEMBL9102311 0.73 CTSK (0.50) CTSKCTSLCTSBELANEHDAC8
SCHEMBL9102306 0.73 CTSK (0.50) CTSKCTSLCTSBELANEHDAC8
SCHEMBL5203085 0.72 HDAC8 (0.51) CTSKCTSLCTSBHDAC8CTSS
SCHEMBL13560013 0.72 HDAC8 (0.43) CTSKCTSLCTSBELANEHDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004071454-A2 SUBSTITUTED AZETIDINE COMPOUNDS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARMACEUTICALS INC. (US) 2004-08-26 WO disclosed