SCHEMBL8312848

SCHEMBL8312848

Oc1ccc2nc(CN3CCC(Cc4ccc(C(F)(F)F)cc4)CC3)[nH]c2c1

nearest known ligand 0.80

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 10/20 0.80
GRIN2B Q13224 10/20 0.80
IDO1 P14902 1/20 0.48
HIF1A Q16665 1/20 0.46
EPAS1 Q99814 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5240925 0.92 GRIN1 (0.67) GRIN1GRIN2BHIF1AEPAS1
SCHEMBL8313704 0.89 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8318042 0.87 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8313723 0.86 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8320273 0.82 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL5241787 0.81 GRIN2B (0.84) GRIN1GRIN2B
SCHEMBL8319076 0.80 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8318192 0.79 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL5269544 0.78 GRIN1 (0.84) GRIN1GRIN2B
SCHEMBL5237195 0.78 GRIN1 (0.84) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048364-A1 2-[(4-BENZYL)-1-PIPERIDINYL)METHYL]BENZIMIDAZOLE-5-OL DERIVATIVES AS NR2B RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2004-06-10 WO disclosed