SCHEMBL8318192

SCHEMBL8318192

Oc1ccc2nc(CN3CCC(Cc4ccccc4F)CC3)[nH]c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 10/20 1.00
GRIN2B Q13224 10/20 1.00
NPC1 O15118 1/20 0.47
GAA P10253 1/20 0.47
DRD4 P21917 1/20 0.47
ATM Q13315 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5239112 0.92 GRIN2B (0.85) GRIN1GRIN2BNPC1GAADRD4
SCHEMBL8319076 0.89 GRIN1 (1.00) GRIN1GRIN2BNPC1GAADRD4
SCHEMBL8313723 0.85 GRIN1 (1.00) GRIN1GRIN2BGAA
SCHEMBL8313704 0.83 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8320273 0.83 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL5240113 0.80 GRIN1 (0.85) GRIN1GRIN2BNPC1GAADRD4
SCHEMBL8318042 0.79 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL8312848 0.79 GRIN1 (0.80) GRIN1GRIN2B
SCHEMBL5237195 0.77 GRIN1 (0.84) GRIN1GRIN2BNPC1GAA
SCHEMBL8313716 0.75 GRIN1 (0.67) GRIN1GRIN2BNPC1GAADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048364-A1 2-[(4-BENZYL)-1-PIPERIDINYL)METHYL]BENZIMIDAZOLE-5-OL DERIVATIVES AS NR2B RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2004-06-10 WO disclosed